SCHEMBL28079083

SCHEMBL28079083

COc1ccc2c(CCNBr)c[nH]c2c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.68
MTNR1B P49286 3/20 0.68
HTR2A P28223 5/20 0.68
MEN1 O00255 4/20 0.66
KMT2A Q03164 4/20 0.66
HTR6 P50406 1/20 0.64
MAPT P10636 2/20 0.59
HPGD P15428 2/20 0.57
MAPK1 P28482 1/20 0.57
GAA P10253 1/20 0.55
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
CYP1A1 P04798 1/20 0.54
MPO P05164 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
HTR1A P08908 1/20 0.54
CYP2D6 P10635 1/20 0.54
NQO2 P16083 1/20 0.54
HTR2B P41595 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12352511 0.87 HTR2A (0.79) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL3816723 0.84 HTR2A (0.73) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL13715395 0.82 HTR2A (0.75) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL9531245 0.81 MTNR1A (0.62) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL30630306 0.81 MTNR1A (1.00) MTNR1AMTNR1BMEN1KMT2AMAPT
SCHEMBL4490583 0.81 MTNR1A (1.00) MTNR1AMTNR1BMEN1KMT2AMAPT
SCHEMBL29874859 0.81 HTR2A (1.00) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL379337 0.81 HTR2A (1.00) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL29899096 0.81 CYP2D6 (0.78) MTNR1AMTNR1BHTR2AMEN1KMT2A
SCHEMBL3812224 0.81 CYP2D6 (0.78) MTNR1AMTNR1BHTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105669525-B A kind of synthetic method of N ((2 (base of 1,3 dioxoisoindolin 2) propiono) 5 methoxyl groups) formamide 苏州艾缇克药物化学有限公司 2018-03-09 CN disclosed
CN-105669525-A Synthetic method of N-((2-(1,3-dioxo-dihydroisoindol-2-yl)-propionyl)-5-methoxy)formamide 苏州艾缇克药物化学有限公司 2016-06-15 CN disclosed