SCHEMBL28079160

SCHEMBL28079160

O=C(O)c1ccc(C(F)(F)I)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 5/20 0.61
RXRA P19793 2/20 0.55
RXRB P28702 2/20 0.55
RXRG P48443 2/20 0.55
TP53 P04637 1/20 0.55
TSHR P16473 1/20 0.55
BCL2L1 Q07817 1/20 0.50
BAD Q92934 1/20 0.50
TPMT P51580 1/20 0.50
EPHX2 P34913 1/20 0.47
PTPN1 P18031 1/20 0.47
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA3 P07451 1/20 0.46
TYR P14679 1/20 0.46
DRD1 P21728 1/20 0.46
CA4 P22748 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28623095 0.84 SRD5A2 (0.57) SRD5A2EPHX2PTPN1CES2CES1
SCHEMBL78879 0.81 SRD5A2 (0.87) SRD5A2RXRARXRBRXRGTP53
SCHEMBL3365796 0.81 TSHR (0.60) SRD5A2TP53TSHRTPMTEPHX2
SCHEMBL4614343 0.81 SRD5A2 (0.65) SRD5A2RXRARXRBRXRGTP53
SCHEMBL1330891 0.81 SRD5A2 (0.87) SRD5A2RXRARXRBRXRGTP53
Terephthalic Acid SCHEMBL28728915 0.80 TSHR (0.67) SRD5A2RXRARXRBRXRGTP53
SCHEMBL505133 0.80 SRD5A2 (0.77) SRD5A2RXRARXRBRXRGBCL2L1
SCHEMBL23521062 0.79 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGTP53
SCHEMBL1042428 0.79 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGTP53
SCHEMBL29208531 0.79 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104341425-B Deuterated acetylene-derivative, its pharmaceutical composition and application 上海医药集团股份有限公司 2018-11-02 CN disclosed
CN-103420977-B There is the acetylene-derivative of anti-tumor activity 上海医药集团股份有限公司 2016-06-22 CN disclosed