SCHEMBL28079302

SCHEMBL28079302

CCN1CCN(Cc2ccc(-c3cccc(C(=O)NC(F)F)c3)cc2C(F)(F)F)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 10/20 0.54
RET P07949 4/20 0.54
KDR P35968 3/20 0.54
STK10 O94804 1/20 0.54
ABL1 P00519 1/20 0.54
BRAF P15056 1/20 0.54
PDGFRA P16234 1/20 0.54
FLT1 P17948 1/20 0.54
CDK11B P21127 1/20 0.54
CDK2 P24941 1/20 0.54
FLT4 P35916 1/20 0.54
FLT3 P36888 1/20 0.54
CDK7 P50613 1/20 0.54
MAPK12 P53778 1/20 0.54
CDK3 Q00526 1/20 0.54
CDK5 Q00535 1/20 0.54
TEK Q02763 1/20 0.54
DDR1 Q08345 1/20 0.54
HIPK1 Q86Z02 1/20 0.54
EPHA2 P29317 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28222510 0.85 RET (0.52) KITRETKDRSTK10ABL1
SCHEMBL12516831 0.80 DDR1 (0.52) KITDDR1MAP3K7MAP4K2MAPK14
Fluoromethane SCHEMBL28079300 0.79 RET (0.47) KITRETKDRSTK10ABL1
SCHEMBL19986834 0.77 HTT (0.54) KITRETKDRDDR1MAP3K7
SCHEMBL14704588 0.77 MAPK14 (0.56) KITRETKDRBRAFDDR1
SCHEMBL27910162 0.76 NR1H2 (0.57) KITRETBRAFCSF1R
SCHEMBL16810188 0.76 DDR1 (0.56) KITRETKDRDDR1ATM
SCHEMBL15121214 0.75 ABL1 (0.59) KITRETKDRSTK10ABL1
SCHEMBL1420613 0.75 CHRM4 (0.67) KITRETKDRSTK10ABL1
SCHEMBL20568827 0.75 EPHA2 (0.63) KITRETKDRSTK10ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103420977-B There is the acetylene-derivative of anti-tumor activity 上海医药集团股份有限公司 2016-06-22 CN disclosed