SCHEMBL2807957

SCHEMBL2807957

Nc1ccc(Br)c(-c2cc(N)ccc2Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
PTPRC P08575 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
KCNH2 Q12809 2/20 0.44
APAF1 O14727 1/20 0.44
TDP2 O95551 1/20 0.44
NSD2 O96028 1/20 0.44
PLA2G1B P04054 1/20 0.44
CTSL P07711 1/20 0.44
HPGD P15428 1/20 0.44
ALOX12 P18054 1/20 0.44
PLCG1 P19174 1/20 0.44
CTSS P25774 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15926831 0.81 ALDH1A1 (0.54) ALDH1A1MEN1KMT2ASMN1; SMN2PTPRC
SCHEMBL29803735 0.81 ALDH1A1 (0.54) ALDH1A1MEN1KMT2ASMN1; SMN2PTPRC
SCHEMBL632670 0.79
SCHEMBL29407502 0.79
SCHEMBL24079298 0.78 HSD17B10 (0.54) ALDH1A1MEN1KMT2ASMN1; SMN2PTPRC
SCHEMBL3088589 0.78 IMPDH2 (0.49) ALDH1A1MEN1KMT2ASMN1; SMN2NPC1
SCHEMBL1503425 0.77 MAPT (0.48) ALDH1A1MEN1KMT2ASMN1; SMN2PTPRC
Methane SCHEMBL28284965 0.77 MAPT (0.48) ALDH1A1MEN1KMT2ASMN1; SMN2PTPRC
SCHEMBL538673 0.77
SCHEMBL29803231 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed
US-6416887-B1 HAVING LAMINATE LAYERS BETWEEN ELECTRODES, USED AS LIGHT SOURCES FOR LIQUID CRYSTAL DISPLAYS KABUSHIKI KAISHA TOYOTA CHUO KENKYUSHO (JP) 2002-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B ALDH1A1 401/4885MEN1 579/4885KMT2A 730/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 ALDH1A1 1480/4885MEN1 379/4885KMT2A 583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.