SCHEMBL28079903

SCHEMBL28079903

O=CC1NN=C(c2ccccc2F)N1C1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.39
HTR2C P28335 4/20 0.39
PLAT P00750 6/20 0.36
MAP4K1 Q92918 1/20 0.35
NISCH Q9Y2I1 1/20 0.34
HTR2B P41595 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
HTR7 P34969 3/20 0.33
HTR1A P08908 1/20 0.33
HTR3A P46098 1/20 0.33
HTR6 P50406 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP3A5 P20815 2/20 0.32
CYP3A7 P24462 2/20 0.32
CYP2C19 P33261 2/20 0.32
PDK4 Q16654 2/20 0.32
CYP3A43 Q9HB55 2/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27770364 0.92 RXFP1 (0.39) HTR2AHTR2CPLATNISCHRXFP1
SCHEMBL27749306 0.77 PTPN11 (0.37) HTR2AHTR2C
SCHEMBL27862115 0.74 PLAT (0.36) PLAT
SCHEMBL28257114 0.73 HTR2C (0.43) HTR2AHTR2CPLATMAP4K1NISCH
SCHEMBL27770358 0.69 PDE4A (0.32)
SCHEMBL16827960 0.65 RXFP1 (0.43) HTR2AHTR2CPLATMAP4K1NISCH
SCHEMBL27272080 0.64 TDP1 (0.34) NISCHRXFP1
SCHEMBL27771646 0.64 HTR2C (0.42) HTR2AHTR2CHTR2B
SCHEMBL16827864 0.63 RXFP1 (0.60) HTR2AHTR2CPLATMAP4K1HTR2B
SCHEMBL13999767 0.61 SCN9A (0.53) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814037-A N1-(3,3,3-trifluoro-2-hydroxo-2-methylpropionyl)-piperidine derivatives as inhibitors of pyruvate dehydrogenase kinase 默克专利股份公司 2016-07-27 CN disclosed