SCHEMBL27770364

SCHEMBL27770364

O=CC1NN=C(c2ccccc2F)N1C1CC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.39
NISCH Q9Y2I1 1/20 0.34
MAPK1 P28482 1/20 0.33
KCNH2 Q12809 1/20 0.33
IL4I1 Q96RQ9 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
PDE6D O43924 5/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
NOTUM Q6P988 2/20 0.30
LMNA P02545 1/20 0.30
PLAT P00750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28079903 0.92 HTR2A (0.39) RXFP1NISCHHTR2AHTR2CPLAT
SCHEMBL27749306 0.84 PTPN11 (0.37) NPC1RAB9ASMN1; SMN2HTR2AHTR2C
SCHEMBL27862115 0.80 PLAT (0.36) PLAT
SCHEMBL27770358 0.75 PDE4A (0.32) MEN1KMT2A
SCHEMBL27770354 0.71 GAA (0.39) NISCHNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL27272080 0.68 TDP1 (0.34) RXFP1NISCHCA1CA2
SCHEMBL28058456 0.66 ALDH1A1 (0.33) LMNA
SCHEMBL27837877 0.66
SCHEMBL28058452 0.64 ALDH1A1 (0.31) LMNA
SCHEMBL28058503 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101495458-B Substituted arylimidazolone and triazolone as inhibitors of vasopressin receptors BAYER IP GMBH 2014-01-29 CN disclosed
CN-101495458-A Substituted arylimidazolone and triazolone as inhibitors of vasopressin receptors BAYER HEALTHCARE AG (DE) 2009-07-29 CN disclosed