SCHEMBL28080023

SCHEMBL28080023

Cc1nc(C2CCCCC2)c(-c2cnccn2)c(C2CCCCC2)n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP11B2 P19099 2/20 0.36
P2RX7 Q99572 4/20 0.35
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CHEK1 O14757 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
PIM1 P11309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3135323 0.69 CYP11B2 (0.47) NPY5RALDH1A1CYP11B2
SCHEMBL28761033 0.69 CYP11B2 (0.47) NPY5RALDH1A1CYP11B2
SCHEMBL4017343 0.68 HDAC3 (0.33) ALDH1A1CYP11B2KDM4EHDAC3HDAC1
SCHEMBL20995461 0.67 CYP11B2 (0.44) NPY5RALDH1A1CYP11B2PIM1
SCHEMBL2355700 0.66 CYP11B2 (0.40) NPY5RALDH1A1CYP11B2HTTKDM4E
SCHEMBL17755587 0.65 PIM1 (0.45) NPY5RHTTRECQLKDM4EHRH3
SCHEMBL17755586 0.65 HTT (0.42) NPY5RHTTRECQLKDM4EHRH3
SCHEMBL548100 0.65 OPRL1 (0.45) ALDH1A1CYP11B2KDM4E
SCHEMBL25419095 0.65 HRH3 (0.34) CYP11B2P2RX7CHEK1CCNA2CDK2
SCHEMBL28197535 0.63 MAP4K4 (0.40) NPY5RCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814022-A Fused bicyclic heteroaromatic derivatives as modulators of tnf activity UCB生物制药私人有限公司 2016-07-27 CN disclosed