SCHEMBL2808025

SCHEMBL2808025

CCC#Cc1cccc(N)c1C

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.48
TSHR P16473 2/20 0.48
PIK3CA P42336 1/20 0.48
ALDH1A1 P00352 6/20 0.41
KDM4E B2RXH2 2/20 0.39
CYP1A2 P05177 2/20 0.39
MAPT P10636 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CD44 P16070 1/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 2/20 0.31
TLR8 Q9NR97 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2806223 0.82 CYP3A4 (0.49) CYP3A4TSHRPIK3CAALDH1A1KDM4E
SCHEMBL3978730 0.82 CYP3A4 (0.55) CYP3A4TSHRPIK3CAALDH1A1KDM4E
SCHEMBL13488446 0.78 PNMT (0.34) CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL2808492 0.78 CYP3A4 (0.54) CYP3A4TSHRPIK3CAALDH1A1KDM4E
SCHEMBL2810978 0.77 TRPA1 (0.43) TSHRALDH1A1MAPTHSD17B10HPGD
SCHEMBL2888201 0.74 KDM4E (0.31) ALDH1A1KDM4EMAPTHSD17B10HPGD
SCHEMBL25654060 0.74 CYP3A4 (0.44) CYP3A4TSHRPIK3CAALDH1A1KDM4E
SCHEMBL2812547 0.73 NPC1 (0.68) CYP3A4TSHRPIK3CAALDH1A1KDM4E
SCHEMBL1507410 0.73 CYP3A4 (0.48) CYP3A4TSHRPIK3CAALDH1A1KDM4E
SCHEMBL19559957 0.73 CYP3A4 (0.45) CYP3A4TSHRALDH1A1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B CYP3A4 1909/4885TSHR 3644/4885PIK3CA 4498/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 CYP3A4 3918/4885TSHR 4692/4885PIK3CA 4324/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.