SCHEMBL28080928

SCHEMBL28080928

Fc1cccnc1OCC(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2B Q13224 2/20 0.44
SSTR4 P31391 2/20 0.43
SCN9A Q15858 1/20 0.42
GPBAR1 Q8TDU6 2/20 0.39
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
HCRTR1 O43613 4/20 0.37
HCRTR2 O43614 4/20 0.37
KCNH2 Q12809 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
P2RY1 P47900 1/20 0.36
ADORA2A P29274 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
FFAR1 O14842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31143575 1.00 RXRA (0.44) RXRAGRIN1GRIN2BSSTR4SCN9A
SCHEMBL18726968 0.82 SCN9A (0.43) SSTR4SCN9AGPBAR1HCRTR1HCRTR2
SCHEMBL16174985 0.79 SSTR4 (0.42) RXRAGRIN1GRIN2BSSTR4SCN9A
SCHEMBL11441604 0.79 SCN9A (0.50) SCN9AGPBAR1HCRTR1HCRTR2KCNH2
SCHEMBL13424282 0.79 SSTR4 (0.45) SSTR4SCN9AGPBAR1HCRTR1HCRTR2
SCHEMBL367912 0.79 L3MBTL1 (0.41) SSTR4SCN9AGPBAR1HCRTR1HCRTR2
SCHEMBL16334635 0.79 SCN9A (0.41) SSTR4SCN9AGPBAR1HCRTR1HCRTR2
SCHEMBL1933518 0.79 SCN9A (0.41) SSTR4SCN9AGPBAR1HCRTR1HCRTR2
SCHEMBL28062293 0.79 SCN9A (0.41) SSTR4SCN9AGPBAR1HCRTR1HCRTR2
SCHEMBL15473322 0.78 CBFB (0.42) RXRAGRIN1GRIN2BSSTR4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104520296-B Pyrrolopyridinone derivatives as TTX-S blocker 拉夸里亚创药株式会社 2016-11-16 CN disclosed