SCHEMBL28080949

SCHEMBL28080949

Cc1ccncc1OCC(F)(F)C(F)F

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.42
HTT P42858 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
CYP17A1 P05093 5/20 0.39
CFTR P13569 4/20 0.39
MAPK1 P28482 2/20 0.37
AAK1 Q2M2I8 4/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28160859 0.83 CYP17A1 (0.51) SSTR4KMT2ACHRNB2CHRNA4CYP17A1
Ammonia Solution, Strong SCHEMBL28408262 0.82 CYP17A1 (0.50) SSTR4KMT2ACHRNB2CHRNA4CYP17A1
SCHEMBL1710086 0.77 KDM4E (0.45) HTTKMT2ASMN1; SMN2CFTRALDH1A1
SCHEMBL16252776 0.76 SSTR4 (0.47) SSTR4CHRNB2CHRNA4CYP17A1AAK1
Ammonia Solution, Strong SCHEMBL28411378 0.76 CYP17A1 (0.50) SSTR4CHRNB2CHRNA4CYP17A1KDM4E
Formic Acid SCHEMBL28012981 0.75 SSTR4 (0.47) SSTR4CHRNB2CHRNA4CYP17A1AAK1
SCHEMBL15350352 0.74 AAK1 (0.37) HTTKMT2ACFTRMAPK1AAK1
Ammonia Solution, Strong SCHEMBL28411555 0.73 CHRNB2 (0.42) SSTR4CHRNB2CHRNA4CYP17A1MAPT
SCHEMBL14424010 0.72 CA12 (0.50) SSTR4HTTKMT2ASMN1; SMN2CHRNB2
SCHEMBL15351760 0.72 AAK1 (0.37) HTTKMT2ASMN1; SMN2CFTRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104520296-B Pyrrolopyridinone derivatives as TTX-S blocker 拉夸里亚创药株式会社 2016-11-16 CN disclosed