Pyrazole

Pyrazole

SCHEMBL28081671

Nc1nc2cc(Cl)c(Cl)cc2s1.c1cn[nH]c1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CYP3A4 P08684 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TSHR P16473 1/20 0.42
CYP2D6 P10635 1/20 0.40
DRD2 P14416 1/20 0.40
PI4KA P42356 4/20 0.39
PI4KB Q9UBF8 4/20 0.39
PIK3CD O00329 4/20 0.39
PIK3CG P48736 4/20 0.39
PIP5K1C O60331 2/20 0.39
MAPT P10636 2/20 0.38
HTT P42858 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
PIK3CA P42336 4/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2899732 0.82 ALDH1A1 (0.59) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
SCHEMBL29462442 0.82 ALDH1A1 (0.59) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
Nitrogen SCHEMBL27684908 0.79 ALDH1A1 (0.55) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
Pyrazole SCHEMBL28081707 0.77 PI4KA (0.46) TP53SMN1; SMN2CYP3A4ALDH1A1PI4KA
SCHEMBL1638626 0.69 AXL (0.53) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
SCHEMBL26927659 0.69 SMN1; SMN2 (0.72) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
SCHEMBL10201412 0.69 ALDH1A1 (0.52) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
SCHEMBL16238119 0.69 SMN1; SMN2 (0.72) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
SCHEMBL29741763 0.69 CYP3A4 (0.53) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR
SCHEMBL21091211 0.69 CYP3A4 (0.53) TP53SMN1; SMN2CYP3A4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105820596-A Tetrahydroquinoline dye, ink and electrowetting display 深圳市国华光电科技有限公司 2016-08-03 CN disclosed