SCHEMBL28082017

SCHEMBL28082017

COc1ccc(COc2ccc(NC(=O)c3cc4cc([N+](=O)[O-])ccc4[nH]3)cc2Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.50
MAPT P10636 5/20 0.49
KMT2A Q03164 5/20 0.49
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 4/20 0.49
MEN1 O00255 4/20 0.49
LMNA P02545 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CYP1A2 P05177 1/20 0.49
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
TDP1 Q9NUW8 1/20 0.48
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
GAA P10253 2/20 0.47
PRNP P04156 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP19A1 P11511 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28832324 0.94 TDP1 (0.49) TP53MAPTKMT2AKDM4EALDH1A1
SCHEMBL28081968 0.91 MAPT (0.49) TP53MAPTKMT2AKDM4EALDH1A1
SCHEMBL28082011 0.90 TDP1 (0.51) MAPTKMT2AKDM4EALDH1A1MEN1
SCHEMBL28081953 0.88 TDP1 (0.48) TDP1PYGLNHERF1
SCHEMBL28257814 0.84 TDP1 (0.51) MAPTKMT2AALDH1A1MEN1LMNA
SCHEMBL28081958 0.84 EGFR (0.51) KMT2AALDH1A1MEN1TDP1PYGL
SCHEMBL28081980 0.84 TP53 (0.69) TP53MAPTKMT2AKDM4EALDH1A1
SCHEMBL28081982 0.83 PYGL (0.56) TP53MAPTKMT2AMEN1LMNA
SCHEMBL28257737 0.83 TDP1 (0.47) TP53MAPTKMT2AKDM4EALDH1A1
SCHEMBL22983913 0.78 MAPT (0.61) MAPTKMT2AALDH1A1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105820104-B A kind of indoles -2- amides compound with anti-inflammatory effect and its application in preparing anti-inflammatory drugs 温州医科大学 2018-12-11 CN disclosed
CN-105820104-A Indole-2-acetamide compound with anti-inflammatory effect, and application thereof in preparation of anti-inflammatory drugs 温州医科大学 2016-08-03 CN disclosed