SCHEMBL28082097

SCHEMBL28082097

[O-][S+](CCCCl)c1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.33
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 3/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP2D6 P10635 3/20 0.32
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
CYP19A1 P11511 2/20 0.31
CYP2E1 P05181 1/20 0.31
CYP2B6 P20813 1/20 0.31
HRH1 P35367 2/20 0.31
CHRNA7 P36544 1/20 0.31
TP53 P04637 1/20 0.31
HTT P42858 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30
CHRM2 P08172 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4681692 0.83 CYP2A6 (0.33) CYP2A6CYP3A4CYP1A2ALDH1A1TDP1
SCHEMBL4681696 0.83 TBXAS1 (0.37) CYP2A6CYP3A4CYP1A2ALDH1A1TDP1
SCHEMBL4684862 0.81 TBXAS1 (0.39) CYP2A6CYP3A4CYP1A2ALDH1A1TDP1
SCHEMBL4684856 0.81 TDP1 (0.33) CYP2A6CYP3A4CYP1A2ALDH1A1TDP1
SCHEMBL4686198 0.80 LMNA (0.33) CYP2A6CYP3A4CYP1A2ALDH1A1TDP1
SCHEMBL4682192 0.80 TBXAS1 (0.41) CYP2A6CYP3A4CYP1A2ALDH1A1HRH1
SCHEMBL4682190 0.80 LMNA (0.33) CYP2A6CYP3A4CYP1A2ALDH1A1TDP1
SCHEMBL4686200 0.80 TBXAS1 (0.41) CYP2A6CYP3A4CYP1A2ALDH1A1HRH1
SCHEMBL4681563 0.79 CYP2A6 (0.35) CYP2A6CYP3A4CYP1A2ALDH1A1CYP2D6
SCHEMBL4681569 0.79 MKNK1 (0.37) CYP2A6CYP3A4CYP1A2ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814054-B Condensed imidazole and pyrazole derivatives as TNF active regulators UCB生物制药私人有限公司 2018-09-25 CN disclosed
CN-105814054-A Fused imidazole and pyrazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed