SCHEMBL28083642

SCHEMBL28083642

CCCC[Sn](CCCC)(CCCC)c1cccc2[nH]ncc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.45
NOS1 P29475 4/20 0.44
AXL P30530 2/20 0.44
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
METAP2 P50579 1/20 0.41
BRD4 O60885 1/20 0.36
DHPS P49366 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
RAF1 P04049 1/20 0.35
BRAF P15056 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RET P07949 1/20 0.35
KIF5B P33176 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10264250 0.71 DRD2 (0.58) IDO1NOS1AXLMETAP2BRD4
SCHEMBL21259457 0.71 IDO1 (0.46) IDO1NOS1AXLMETAP2
SCHEMBL1453289 0.70 HTR1B (0.40) ALDH1A1NPC1HTTRAB9A
SCHEMBL691687 0.70 LMNA (0.49) MAPTALDH1A1LMNACYP1A2CYP3A4
SCHEMBL29416223 0.69 IDO1 (0.51) IDO1NOS1AXLJAK2JAK1
SCHEMBL12166325 0.69 IDO1 (0.51) IDO1NOS1AXLJAK2JAK1
SCHEMBL28358722 0.69 KDM4E (0.42) IDO1ALDH1A1NPC1LMNACYP1A2
SCHEMBL2633084 0.68 IDO1 (0.55) IDO1NOS1AXLJAK2JAK1
SCHEMBL691136 0.68 KDM4E (0.41) POLBMAPTALDH1A1NPC1LMNA
SCHEMBL24652885 0.68 IDO1 (0.48) IDO1NOS1AXLJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829308-B Isochromene derivatives as phosphoinositide 3-kinase inhibitors 奇斯药制品公司 2019-03-08 CN disclosed
CN-105829308-A Isochromene derivatives as phosphoinositide 3-kinase inhibitors 奇斯药制品公司 2016-08-03 CN disclosed