SCHEMBL28083786

SCHEMBL28083786

Cc1c(C(=O)O)cccc1C(=O)O.N#CC#N.c1ccc(-n2cccn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
HDAC4 P56524 1/20 0.41
PPARG P37231 2/20 0.41
PPARA Q07869 2/20 0.41
KAT6A Q92794 2/20 0.40
ELANE P08246 1/20 0.40
NOTUM Q6P988 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2C9 P11712 1/20 0.38
DGAT1 O75907 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28840375 0.94 LMNA (0.46) LMNAHDAC4PPARGPPARAKAT6A
SCHEMBL15524867 0.79 MYC (0.45) LMNAELANEKDM4EALDH1A1MAPK1
Bicarbonate SCHEMBL10672835 0.77 NOTUM (0.57) LMNAHDAC4KAT6ANOTUMKDM4E
SCHEMBL27312206 0.77 TSHR (0.53) LMNAKDM4EALDH1A1MAPTMEN1
SCHEMBL27605945 0.75 LMNA (0.47) LMNAHDAC4KAT6AELANEALDH1A1
SCHEMBL27250 0.73 NOTUM (0.65) LMNAHDAC4KAT6ANOTUMKDM4E
SCHEMBL27584512 0.73 LMNA (0.48) LMNAHDAC4KAT6ANOTUMKDM4E
SCHEMBL28803951 0.73 LMNA (0.42) LMNAHDAC4KAT6AELANENOTUM
SCHEMBL1586230 0.73 ELANE (0.49) LMNAKAT6AELANEKDM4EALDH1A1
Methylamine SCHEMBL27947262 0.72 NOTUM (0.59) LMNAHDAC4KAT6ANOTUMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103833744-B 1 ethyl pyrazolyl acrylonitrile compound and application thereof 沈阳中化农药化工研发有限公司 2016-12-21 CN disclosed
CN-103833668-B O-trifluoromethyl phenylpropen nitrile compounds and application thereof 沈阳中化农药化工研发有限公司 2016-08-03 CN disclosed