SCHEMBL28084147

SCHEMBL28084147

N#Cc1ccc(CNC(=O)[C@@H](N)Cc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSC P53634 2/20 0.56
SLC1A3 P43003 1/20 0.52
SLC1A2 P43004 1/20 0.52
EGFR P00533 2/20 0.49
TPH1 P17752 1/20 0.49
SRC P12931 1/20 0.49
MMP8 P22894 1/20 0.49
ALPI P09923 1/20 0.47
PKM P14618 1/20 0.47
PTGS1 P23219 1/20 0.47
XIAP P98170 1/20 0.47
SLC7A5 Q01650 1/20 0.47
BACE1 P56817 1/20 0.46
BACE2 Q9Y5Z0 1/20 0.46
MMP2 P08253 1/20 0.46
MAOA P21397 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28084151 1.00 CTSC (0.56) CTSCSLC1A3SLC1A2EGFRTPH1
Hydrochloric Acid SCHEMBL14486038 0.99 CTSC (0.54) CTSCSLC1A3SLC1A2EGFRTPH1
Hydrochloric Acid SCHEMBL14486037 0.99 CTSC (0.54) CTSCSLC1A3SLC1A2EGFRTPH1
SCHEMBL15307625 0.89 LOXL2 (0.57) CTSCSLC1A3SLC1A2TPH1
SCHEMBL7413310 0.87 ALPI (0.61) CTSCEGFRSRCMMP8ALPI
SCHEMBL3114367 0.87 ALPI (0.61) CTSCEGFRSRCMMP8ALPI
SCHEMBL17366111 0.87 MMP8 (0.51) CTSCSLC1A3SLC1A2EGFRSRC
Hydrochloric Acid SCHEMBL3385081 0.85 MMP8 (0.59) CTSCEGFRSRCMMP8ALPI
Hydrochloric Acid SCHEMBL27492563 0.85 MMP8 (0.59) CTSCEGFRSRCMMP8ALPI
SCHEMBL6440952 0.85 MMP8 (0.61) SLC1A3SLC1A2MMP8MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103687846-B Benzyl amine derivative as inhibitors of plasma kallikrein 卡尔维斯塔制药有限公司 2016-06-22 CN disclosed