SCHEMBL28085472

SCHEMBL28085472

COc1ccc(Oc2ccc(OB(O)O)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.58
CA1 P00915 5/20 0.52
CA2 P00918 5/20 0.52
ENPP2 Q13822 2/20 0.52
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA12 O43570 1/20 0.50
CA14 Q9ULX7 1/20 0.50
PARP10 Q53GL7 1/20 0.48
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ACHE P22303 1/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
ESR2 Q92731 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MAPK1 P28482 2/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL351810 0.93 CA1 (0.58) LTA4HCA1CA2ENPP2CA7
SCHEMBL28085474 0.85 SMN1; SMN2 (0.61) LTA4HENPP2ALDH1A1MEN1KMT2A
SCHEMBL29141449 0.83 CA1 (0.48) LTA4HCA1CA2ENPP2CA7
SCHEMBL28600111 0.81 CA1 (0.52) LTA4HCA1CA2ENPP2CA7
SCHEMBL3800806 0.80 CA1 (0.38) CA1CA2ENPP2CA7CA9
SCHEMBL166536 0.80 CA1 (0.79) LTA4HCA1CA2CA7CA9
SCHEMBL11580995 0.80 CA1 (0.79) LTA4HCA1CA2CA7CA9
SCHEMBL83811 0.80 CA1 (0.79) LTA4HCA1CA2CA7CA9
SCHEMBL2762065 0.79 CA1 (0.61) LTA4HCA1CA2CA9PARP10
SCHEMBL6661512 0.78 IDO1 (0.50) CA1CA2ENPP2HTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106279172-A Purinone compound as inhibitors of kinases 药品循环有限责任公司 2017-01-04 CN disclosed
CN-104640861-B Purinone compounds as kinase inhibitors 药品循环公司 2016-08-24 CN disclosed
CN-104844609-B The irreversible bruton's tyrosine kinase inhibitor of dibit point 杭州和正医药有限公司 2016-07-13 CN disclosed