SCHEMBL28085556

SCHEMBL28085556

COc1ccc(CNc2ncccc2C=O)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.62
EGFR P00533 2/20 0.49
POLB P06746 1/20 0.49
NR2F2 P24468 1/20 0.49
HIF1A Q16665 1/20 0.48
CCNB2 O95067 1/20 0.45
CDK1 P06493 1/20 0.45
CCNB1 P14635 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
CCNB3 Q8WWL7 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPT P10636 1/20 0.45
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
APP P05067 1/20 0.44
VNN1 O95497 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29957028 0.83 EGFR (0.50) NPC1EGFRNR2F2HIF1AMEN1
SCHEMBL19641368 0.83 NPC1 (0.51) NPC1EGFRPOLBNR2F2CCNB2
SCHEMBL27787171 0.82 KDM4E (0.51) EGFRPOLBKMT2AMAPTHPGD
SCHEMBL19641279 0.82 NPC1 (0.50) NPC1EGFRPOLBNR2F2CCNB2
SCHEMBL12675591 0.80 NPC1 (0.64) NPC1EGFRPOLBNR2F2HIF1A
SCHEMBL28283742 0.80 NPC1 (0.64) NPC1EGFRPOLBNR2F2HIF1A
SCHEMBL8835483 0.79 RAB9A (0.60) NPC1MEN1KMT2AMAPTLMNA
SCHEMBL21382408 0.79 NPC1 (0.62) NPC1EGFRPOLBNR2F2HIF1A
SCHEMBL6131117 0.79 NPC1 (0.62) NPC1EGFRPOLBNR2F2HIF1A
SCHEMBL1347342 0.79 NPC1 (0.62) NPC1EGFRPOLBNR2F2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106220623-A Compounds and methods for and indication thereof for kinases regulation 普莱希科公司 2016-12-14 CN disclosed
CN-102947305-B Compounds and methods for kinase modulation and indications therefor 普莱希科公司 2016-07-06 CN disclosed