Oxeladin

Oxeladin

SCHEMBL28086122

CCN(CC)CCOCCOC(=O)C(CC)(CC)c1ccccc1.CCN(CC)CCc1nc(-c2ccccc2)no1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.60
CYP2D6 P10635 3/20 0.60
HIF1A Q16665 1/20 0.60
HTR1A P08908 1/20 0.60
HRH3 Q9Y5N1 1/20 0.60
CHRM2 P08172 3/20 0.46
CHRM1 P11229 3/20 0.46
CHRM3 P20309 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
LMNA P02545 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
SCN1A P35498 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxeladin SCHEMBL405413 0.83 CHRM2 (0.64) CYP1A2CYP2D6HIF1ACHRM2CHRM1
Oxolamine SCHEMBL4414451 0.80 CYP1A2 (0.78) CYP1A2CYP2D6HIF1AHTR1AHRH3
SCHEMBL3366202 0.80 CHRM2 (0.56) CYP1A2CYP2D6CHRM2CHRM1CHRM3
Carbetapentane SCHEMBL13724360 0.78 CHRM2 (0.71) CYP1A2CYP2D6HIF1AHTR1AHRH3
Oxolamine SCHEMBL893333 0.78 HTR1A (1.00) CYP1A2CYP2D6HIF1AHTR1AHRH3
Oxolamine SCHEMBL1652318 0.76 HTR1A (0.97) CYP1A2CYP2D6HIF1AHTR1AHRH3
Oxolamine SCHEMBL3498928 0.76 CYP1A2 (1.00) CYP1A2CYP2D6HIF1AHTR1AHRH3
Oxeladin SCHEMBL405412 0.76 CYP2D6 (0.62) CYP1A2CYP2D6HIF1ACHRM2CHRM1
SCHEMBL3362813 0.75 CHRM2 (0.51) CYP1A2CYP2D6CHRM2CHRM1CHRM3
SCHEMBL3364929 0.73 CHRM2 (0.49) CYP1A2CYP2D6CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed