Penthienate

Penthienate

SCHEMBL28086303

CCCN.CC[N+](C)(CC)CCOC(=O)C(O)(c1cccs1)C1CCCC1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 11/20 0.62
CHRM2 P08172 10/20 0.62
SLC6A3 Q01959 1/20 0.62
KCNH2 Q12809 1/20 0.62
CHRM3 P20309 10/20 0.62
CHRM4 P08173 3/20 0.62
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
LMNA P02545 1/20 0.44
SCN1A P35498 2/20 0.42
SCN2A Q99250 2/20 0.42
SCN3A Q9NY46 2/20 0.42
POLB P06746 1/20 0.39
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Penthienate SCHEMBL31393386 0.95 CHRM1 (0.68) CHRM1CHRM2SLC6A3KCNH2CHRM3
Penthienate SCHEMBL250881 0.94 CHRM1 (0.67) CHRM1CHRM2SLC6A3KCNH2CHRM3
SCHEMBL15095409 0.81 CHRM2 (0.62) CHRM1CHRM2SLC6A3KCNH2CHRM3
SCHEMBL2795158 0.79 CHRM2 (0.73) CHRM1CHRM2SLC6A3KCNH2CHRM3
Oxyphenonium SCHEMBL250615 0.77 CHRM2 (1.00) CHRM1CHRM2SLC6A3KCNH2CHRM3
Oxyphenonium SCHEMBL250614 0.77 CHRM2 (1.00) CHRM1CHRM2SLC6A3KCNH2CHRM3
Oxyphenonium SCHEMBL2030870 0.76 CHRM2 (0.98) CHRM1CHRM2SLC6A3KCNH2CHRM3
Oxyphenonium SCHEMBL248890 0.76 CHRM2 (0.98) CHRM1CHRM2SLC6A3KCNH2CHRM3
Penthienate SCHEMBL5886141 0.76 CHRM1 (0.49) CHRM1CHRM2SLC6A3KCNH2CHRM3
SCHEMBL1234853 0.74 CHRM3 (0.63) CHRM1CHRM2CHRM3CHRM4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed