SCHEMBL28086633

SCHEMBL28086633

CC(Nc1ccc2nc[nH]c2c1)C1CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.44
ADRA2A P08913 1/20 0.43
ADRA2C P18825 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
QPCT Q16769 12/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 2/20 0.41
HTT P42858 1/20 0.41
CDK1 P06493 2/20 0.40
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17036636 0.77 ADRA2A (0.54) EPHX1ADRA2AADRA2CADRA1DADRA1A
SCHEMBL18649372 0.75 ADRA2A (0.51) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL3597855 0.72 PRKCI (0.41) EPHX1QPCTSMN1; SMN2POLBHTT
SCHEMBL11557199 0.70 NAMPT (0.52) EPHX1ADRA2AADRA2CADRA1DADRA1A
SCHEMBL2545182 0.70 EPHX1 (0.48) EPHX1ADRA2AADRA2CADRA1DADRA1A
SCHEMBL2544250 0.70 QPCT (0.67) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL5063947 0.69 ADRA2A (0.58) EPHX1ADRA2AADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL7093142 0.69 ROCK1 (0.48) HTTCDK1TP53
SCHEMBL29399373 0.69 QDPR (0.47) EPHX1QPCTNPC1MAPT
SCHEMBL1080493 0.69 NPC1 (0.41) EPHX1QPCTSMN1; SMN2POLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103992310-B One group replaces benzo heterocyclic amine derivant and preparation method thereof and the related application as IMPDH inhibitor 中国医学科学院医药生物技术研究所 2016-07-06 CN disclosed