SCHEMBL28087712

SCHEMBL28087712

CC(C)(C)OC(=O)Nc1ccc2c(cnn2C(=O)OC(C)(C)C)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.55
ITK Q08881 1/20 0.55
ROCK2 O75116 3/20 0.52
ROCK1 Q13464 2/20 0.52
CHEK2 O96017 1/20 0.52
PRKACA P17612 1/20 0.52
RPS6KA3 P51812 1/20 0.52
PAK1 Q13153 1/20 0.52
DYRK1A Q13627 1/20 0.52
PRKD2 Q9BZL6 1/20 0.52
TAOK1 Q7L7X3 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
EEF2K O00418 1/20 0.52
MAP4K4 O95819 1/20 0.52
CLK2 P49760 1/20 0.52
GSK3B P49841 1/20 0.52
PRKX P51817 1/20 0.52
NEK4 P51957 1/20 0.52
PRKG2 Q13237 1/20 0.52
PKN2 Q16513 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28087693 0.90 EGFR (0.46) EGFRITKROCK2ROCK1CHEK2
SCHEMBL6342427 0.88 EGFR (0.51) EGFRITKROCK2ROCK1CHEK2
SCHEMBL18136169 0.85 ACSS2 (0.44) EGFRITKDYRK1AGSK3BACSS2
SCHEMBL16406932 0.85 NOTUM (0.54) DYRK1AGSK3BRAB9ANPC1ACSS2
SCHEMBL16938553 0.83 ROCK2 (0.52) EGFRITKROCK2ROCK1CHEK2
SCHEMBL16455688 0.82 ROCK2 (0.50) EGFRITKROCK2ROCK1CHEK2
SCHEMBL12692642 0.81 TAOK1 (0.46) EGFRITKROCK2ROCK1CHEK2
SCHEMBL23266477 0.80 HDAC8 (0.51) EGFRITKROCK2ROCK1CHEK2
SCHEMBL31414297 0.80 ROCK2 (0.49) EGFRITKROCK2ROCK1CHEK2
SCHEMBL13539429 0.80 SLC22A12 (0.52) EGFRITKROCK2ROCK1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106170486-A Novel indazolecarboxamides, method for the production thereof, pharmaceutical preparations containing the same and use thereof for producing medicaments 拜耳医药股份有限公司 2016-11-30 CN disclosed