SCHEMBL28088013

SCHEMBL28088013

Fc1c(-c2ccccc2)oc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
CYP3A4 P08684 3/20 0.53
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
KDM4E B2RXH2 2/20 0.53
LMNA P02545 2/20 0.53
CA12 O43570 2/20 0.53
TP53 P04637 2/20 0.53
ABCB1 P08183 2/20 0.53
AR P10275 2/20 0.53
CYP1B1 Q16678 2/20 0.53
CA9 Q16790 2/20 0.53
ADORA3 P0DMS8 2/20 0.53
ALOX15 P16050 2/20 0.53
MAPK1 P28482 2/20 0.53
DDR2 Q16832 1/20 0.53
CALM1 P0DP23 1/20 0.53
PKM P14618 1/20 0.53
ABCG2 Q9UNQ0 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28212030 0.88 MAPK14 (0.55) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL31098999 0.85 KMT2A (0.65) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL28088011 0.85 LMNA (0.58) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL28088149 0.85 TNKS (0.49) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL28088260 0.82 CYP3A4 (0.54) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL28088009 0.81 ABCG2 (0.64) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL28195347 0.79 CYP3A4 (0.53) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL592430 0.77 CA1 (0.55) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL28139718 0.76 ELANE (0.44) KMT2AMEN1CYP3A4CA1CA2
SCHEMBL13955890 0.75 CYP3A4 (0.53) KMT2AMEN1CYP3A4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105837539-B Method for substituting 2-site aryl for 3-site fluoro of benzofuran ring 复旦大学 2018-11-13 CN disclosed
CN-105837539-A Method for substituting 2-site aryl for 3-site fluoro of benzofuran ring 复旦大学 2016-08-10 CN disclosed