SCHEMBL28088258

SCHEMBL28088258

COc1cccc(-c2oc3ccccc3c2F)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.64
CYP3A4 P08684 6/20 0.64
HPGD P15428 6/20 0.64
MAPT P10636 5/20 0.64
TSHR P16473 5/20 0.64
KMT2A Q03164 4/20 0.64
TP53 P04637 3/20 0.64
CYP2C9 P11712 3/20 0.64
CYP2C19 P33261 3/20 0.64
MEN1 O00255 3/20 0.64
MAPK1 P28482 3/20 0.64
CYP2D6 P10635 2/20 0.64
TDP1 Q9NUW8 2/20 0.64
ALOX12 P18054 1/20 0.64
SMN1; SMN2 Q16637 3/20 0.50
CSNK2A2 P19784 1/20 0.50
CSNK2B P67870 1/20 0.50
CSNK2A1 P68400 1/20 0.50
ALDH1A1 P00352 6/20 0.49
HSD17B10 Q99714 5/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7527814 0.84 KDM4E (0.65) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL28088009 0.83 ABCG2 (0.64) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL4649960 0.80 KDM4E (0.76) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL29519168 0.78 KDM4E (0.73) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL30667386 0.78 KDM4E (1.00) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL4649962 0.78 KDM4E (1.00) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL6129737 0.78 KDM4E (0.73) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL28088013 0.77 KMT2A (0.53) KDM4ECYP3A4HPGDMAPTKMT2A
SCHEMBL23373166 0.77 KDM4E (0.57) KDM4ECYP3A4HPGDMAPTTSHR
SCHEMBL12203173 0.76 NPC1 (0.59) KDM4ECYP3A4HPGDMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105837539-A Method for substituting 2-site aryl for 3-site fluoro of benzofuran ring 复旦大学 2016-08-10 CN disclosed