SCHEMBL28089016

SCHEMBL28089016

FC(F)(F)On1nnc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
KMT2A Q03164 5/20 0.47
SLC9A1 P19634 3/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 1/20 0.46
MAPK1 P28482 1/20 0.46
ATM Q13315 1/20 0.46
KEAP1 Q14145 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
THPO P40225 1/20 0.46
CYP4Z1 Q86W10 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8227040 0.81 TSHR (0.53) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL21104745 0.79 TSHR (0.58) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL736439 0.78 TSHR (0.61) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL29389351 0.78 TSHR (0.61) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL16497703 0.78 TSHR (0.53) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL31483487 0.76 TSHR (0.59) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL17110689 0.76 TSHR (0.59) TSHRNPSR1RXFP1KMT2ASLC9A1
SCHEMBL22954104 0.76 PKM (0.47) MAPK1GRM2
SCHEMBL30668172 0.76 PKM (0.47) MAPK1GRM2
SCHEMBL26231886 0.76 ALDH1A1 (0.36) NPSR1KMT2AMAPTPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102272105-B enantiomerically enriched aryloazol-2-yl cyanoethylamino parasiticidal compounds 梅瑞尔公司 2016-09-14 CN disclosed