SCHEMBL28089129

SCHEMBL28089129

CN1C=Cc2ccccc2C1C=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.49
CCL2 P13500 1/20 0.49
ATM Q13315 1/20 0.36
CYP3A4 P08684 3/20 0.33
HTR2A P28223 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
ALDH1A1 P00352 6/20 0.33
MAPT P10636 4/20 0.33
KDM4E B2RXH2 4/20 0.31
LMNA P02545 2/20 0.31
TP53 P04637 1/20 0.31
CHRM2 P08172 1/20 0.31
CYP2D6 P10635 1/20 0.31
CHRM1 P11229 1/20 0.31
DRD2 P14416 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
NFKB1 P19838 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27913881 0.98 BRD4 (0.47) BRD4CCL2ATMCYP3A4HTR2A
SCHEMBL27682027 0.80 BRD4 (0.40) BRD4CCL2ATMCYP3A4HTR2A
SCHEMBL28089132 0.80 BRD4 (0.33) BRD4CCL2SLC6A2SLC6A3
SCHEMBL28089151 0.80 KDM4E (0.36) BRD4CCL2ALDH1A1KDM4E
SCHEMBL28507942 0.78 BRD4 (0.32) BRD4CCL2ALDH1A1
SCHEMBL28001004 0.78 CHEK1 (0.33) BRD4CCL2RET
SCHEMBL28089286 0.78 ADORA3 (0.33) BRD4CCL2
SCHEMBL28824445 0.78 BRD4 (0.40) BRD4CCL2ATMHTR2AALDH1A1
Hydrochloric Acid SCHEMBL27896263 0.78 BRD4 (0.40) BRD4CCL2ATMCYP3A4HTR2A
SCHEMBL28089255 0.78 KDM4E (0.36) BRD4CCL2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105828820-A Bromodomain inhibitors 赛尔基因昆蒂赛尔研究公司 2016-08-03 CN disclosed