SCHEMBL28089255

SCHEMBL28089255

CN1C=Cc2cc(F)ccc2C1C=O

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
BRD4 O60885 11/20 0.32
CCL2 P13500 9/20 0.32
SRD5A1 P18405 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28089151 0.89 KDM4E (0.36) KDM4EALDH1A1BRD4CCL2
SCHEMBL28089132 0.83 BRD4 (0.33) BRD4CCL2
SCHEMBL28043653 0.81 BRD4 (0.35) BRD4CCL2
SCHEMBL28507942 0.81 BRD4 (0.32) ALDH1A1BRD4CCL2SRD5A1
SCHEMBL28089129 0.78 BRD4 (0.49) KDM4EALDH1A1BRD4CCL2
Hydrochloric Acid SCHEMBL27913881 0.77 BRD4 (0.47) KDM4EALDH1A1BRD4CCL2
SCHEMBL28001004 0.75 CHEK1 (0.33) BRD4CCL2
SCHEMBL28089257 0.73 ERN1 (0.39) BRD4
SCHEMBL28089286 0.72 ADORA3 (0.33) BRD4CCL2
SCHEMBL27707872 0.66 CHRNB2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105828820-A Bromodomain inhibitors 赛尔基因昆蒂赛尔研究公司 2016-08-03 CN disclosed