SCHEMBL2808939

SCHEMBL2808939

Oc1nc(O)c2cnn(-c3cc(Cl)ccc3Cl)c2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 1/20 0.47
THRB P10828 1/20 0.45
HTT P42858 1/20 0.39
ESR1 P03372 1/20 0.39
KDM4E B2RXH2 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GRM1 Q13255 4/20 0.37
TP53 P04637 3/20 0.36
GRM5 P41594 2/20 0.36
LMNA P02545 2/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
JAK3 P52333 1/20 0.35
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 1/20 0.34
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2786952 0.83 ALDH1A1 (0.48) PDE9AGRM1GRM5LMNAALDH1A1
SCHEMBL2807304 0.77 PDE9A (0.48) PDE9ATHRBHTTESR1KDM4E
SCHEMBL2788919 0.70 GRM1 (0.50) HTTKDM4EGRM1GRM5LMNA
SCHEMBL13790292 0.69 ALDH1A1 (0.46) PDE9AGRM1GRM5LMNAALDH1A1
SCHEMBL31341738 0.69 CYP17A1 (0.38) PDE9ASMN1; SMN2MAPT
SCHEMBL1750717 0.68 HTT (0.43) PDE9ATHRBHTTESR1KDM4E
SCHEMBL13087861 0.65 SMN1; SMN2 (0.55) HTTKDM4EL3MBTL1TP53LMNA
SCHEMBL7953211 0.65 CDK4 (0.56) THRBKDM4EL3MBTL1GRM1GRM5
SCHEMBL1751055 0.65 ESR1 (0.42) PDE9ATHRBHTTESR1KDM4E
SCHEMBL1457129 0.64 PDE9A (1.00) PDE9ACDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118367-A2 ANTIVIRAL PYRIMIDINES PROGENICS PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed