SCHEMBL28089438

SCHEMBL28089438

CCC(=O)Nc1cccc(N2CCNCC2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.55
ITGA2B P08514 1/20 0.55
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
POLB P06746 2/20 0.54
KDM4E B2RXH2 1/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
BLM P54132 1/20 0.54
CHEK1 O14757 1/20 0.54
AURKA O14965 1/20 0.54
DAPK3 O43293 1/20 0.54
JAK2 O60674 1/20 0.54
PRKD3 O94806 1/20 0.54
PAK4 O96013 1/20 0.54
ABL1 P00519 1/20 0.54
NTRK1 P04629 1/20 0.54
LCK P06239 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1383637 0.85 GAA (0.56) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL10396194 0.84 POLB (0.56) MEN1KMT2APOLBKDM4EUSP2
Hydrochloric Acid SCHEMBL3976781 0.83 GAA (0.54) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL532030 0.83 HTT (0.73) ITGB3ITGA2BMEN1KMT2APOLB
SCHEMBL8576378 0.83 POLB (0.56) MEN1KMT2APOLBKDM4EUSP2
SCHEMBL12913021 0.82 ADRB1 (0.56) MEN1KMT2APOLBKDM4EUSP2
SCHEMBL14365681 0.82 CNR1 (0.53) MEN1KMT2APOLBKDM4EUSP2
Hydrochloric Acid SCHEMBL6528621 0.82 HTR6 (0.58) MEN1KMT2APOLBKDM4EUSP2
SCHEMBL22169762 0.81 MAPT (0.52) POLBALDH1A1MAPTJAK2HTT
SCHEMBL1382777 0.81 ABL1 (0.57) ITGB3ITGA2BMEN1KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849096-B Piperidine derivatives having multimodal activity against pain 埃斯蒂文制药股份有限公司 2019-11-29 CN disclosed
CN-105849096-A Piperidine derivatives having multimodal activity against pain 埃斯蒂文博士实验室股份有限公司 2016-08-10 CN disclosed