SCHEMBL28089629

SCHEMBL28089629

COCC(=O)Nc1ccccc1Br

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.68
GAA P10253 1/20 0.60
ALDH1A1 P00352 4/20 0.60
KDM4E B2RXH2 1/20 0.57
HSD17B10 Q99714 1/20 0.57
L3MBTL1 Q9Y468 5/20 0.57
TDP1 Q9NUW8 3/20 0.57
HPGD P15428 2/20 0.56
LMNA P02545 2/20 0.53
MAPK1 P28482 2/20 0.53
CYP2C19 P33261 1/20 0.53
MAPT P10636 1/20 0.53
ALOX12 P18054 1/20 0.53
HTT P42858 1/20 0.53
KMT2A Q03164 1/20 0.53
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27144018 0.81 TSHR (0.70) TSHRGAAALDH1A1KDM4EHSD17B10
SCHEMBL7547745 0.81 SMN1; SMN2 (0.71) TSHRGAAALDH1A1KDM4EHSD17B10
SCHEMBL6361102 0.80 KMT2A (0.57) ALDH1A1L3MBTL1TDP1LMNAMAPK1
SCHEMBL19388071 0.79 POLB (0.68) TSHRGAAALDH1A1KDM4EHSD17B10
SCHEMBL11718177 0.79 TSHR (0.68) TSHRGAAKDM4EHSD17B10HPGD
SCHEMBL31656350 0.79 TSHR (0.68) TSHRGAAALDH1A1KDM4EHSD17B10
SCHEMBL14818749 0.79 TSHR (0.68) TSHRGAAALDH1A1KDM4EHSD17B10
SCHEMBL1116453 0.79 LMNA (0.58) ALDH1A1L3MBTL1TDP1LMNAMAPK1
SCHEMBL5360905 0.78 L3MBTL1 (0.58) ALDH1A1L3MBTL1TDP1HPGDLMNA
SCHEMBL1189089 0.78 HTT (0.55) GAAALDH1A1HSD17B10L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777756-B Heteroaryl compound and its application in drug 广东东阳光药业有限公司 2019-03-01 CN disclosed
CN-105777756-A Heteroaryl compound and application thereof in medicines 广东东阳光药业有限公司 2016-07-20 CN disclosed