SCHEMBL28090478

SCHEMBL28090478

CC(C)(C)C(=O)ONc1ccccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PDK3 Q15120 1/20 0.46
PDK4 Q16654 1/20 0.46
HTT P42858 4/20 0.41
KMT2A Q03164 3/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 2/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.38
ALDH1A1 P00352 2/20 0.38
ATM Q13315 1/20 0.38
ELANE P08246 1/20 0.38
EGFR P00533 1/20 0.37
CETP P11597 1/20 0.37
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28832949 0.79 PDK1 (0.51) PDK1PDK2PDK3PDK4HTT
SCHEMBL28876956 0.77 POLB (0.49) KMT2ARAB9AMEN1NPC1LMNA
SCHEMBL1925308 0.76 MAPT (0.45) ELANEMAPT
SCHEMBL2909082 0.73 PDK1 (0.68) PDK1PDK2PDK3PDK4HTT
SCHEMBL30806792 0.73 PDK1 (0.68) PDK1PDK2PDK3PDK4HTT
SCHEMBL10192394 0.70 ELANE (0.57) KMT2ARAB9ANPC1L3MBTL1ALDH1A1
SCHEMBL19280535 0.69 PDK1 (0.68) PDK1PDK2PDK3PDK4HTT
SCHEMBL28869670 0.69 ELANE (0.62) LMNAELANEMAPT
SCHEMBL30976363 0.69 PDK1 (0.54) PDK1PDK2PDK3PDK4HTT
SCHEMBL632629 0.69 PDK1 (0.54) PDK1PDK2PDK3PDK4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777667-A Preparation method of anti-depression drug 1-[2-(2,4-dimethylphenylthio)phenyl]piperazine 康普药业股份有限公司 2016-07-20 CN disclosed