SCHEMBL28090546

SCHEMBL28090546

COc1cc(C)c(-n2ccnc2)cc1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.48
CYP11B2 P19099 2/20 0.48
CYP19A1 P11511 1/20 0.48
ALDH1A1 P00352 5/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CGAS Q8N884 1/20 0.41
MAPT P10636 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
POLB P06746 1/20 0.38
LMNA P02545 2/20 0.37
FGFR1 P11362 1/20 0.37
HPGD P15428 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28003336 0.80 EGLN2 (0.37) CYP11B1CYP11B2CYP19A1ALDH1A1LMNA
SCHEMBL28090553 0.80 CYP19A1 (0.51) CYP11B1CYP11B2CYP19A1ALDH1A1TSHR
SCHEMBL7738817 0.77 CYP11B1 (0.65) CYP11B1CYP11B2CYP19A1ALDH1A1TSHR
SCHEMBL29205321 0.76 ALDH1A1 (0.54) CYP11B1CYP11B2CYP19A1ALDH1A1CGAS
SCHEMBL6540845 0.76 CYP11B1 (0.54) CYP11B1CYP11B2CYP19A1ALDH1A1MAPT
SCHEMBL29105016 0.75 IDO1 (0.47) CYP11B1CYP11B2CYP19A1ALDH1A1TDP1
SCHEMBL1239793 0.74 ALDH1A1 (0.59) CYP11B1CYP11B2CYP19A1ALDH1A1TSHR
SCHEMBL1239502 0.73 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1ALDH1A1TSHR
SCHEMBL8076637 0.71 ALDH1A1 (0.68) ALDH1A1TSHRKDM4ETDP1MAPT
SCHEMBL29205323 0.71 ALDH1A1 (0.50) CYP11B1CYP11B2CYP19A1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104529809-B A kind of preparation method of polysubstituted imidazole derivative 浙江大学 2016-08-24 CN disclosed