SCHEMBL28090559

SCHEMBL28090559

COc1ccc(-n2ncc(C(=O)c3ccccc3)n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.55
ADORA2A P29274 1/20 0.51
ADORA1 P30542 1/20 0.51
HTT P42858 2/20 0.48
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
ALDH1A1 P00352 3/20 0.46
GAA P10253 1/20 0.46
KDM4E B2RXH2 2/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RPA1 P27694 1/20 0.45
HSD11B1 P28845 1/20 0.44
KCNA5 P22460 1/20 0.43
ABCG2 Q9UNQ0 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28090836 0.85 HDAC1 (0.51) MAPK14ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL15577134 0.84 ALDH1A1 (0.51) MAPK14ADORA2AADORA1HTTALDH1A1
SCHEMBL28090523 0.82 MAPT (0.44) ADORA2AADORA1HTTCES2CES1
SCHEMBL28090835 0.82 HTT (0.47) MAPK14ADORA2AADORA1HTTALDH1A1
SCHEMBL28090831 0.82 MAPK14 (0.52) MAPK14ALDH1A1KDM4ELMNAMEN1
SCHEMBL28090834 0.78 HDAC1 (0.49) MAPK14ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL28090875 0.77 ALDH1A1 (0.69) MAPK14ADORA2AADORA1HTTCES2
SCHEMBL23354751 0.76 PDE4D (0.54) HTTALDH1A1GAAKDM4ENPC1
SCHEMBL29873885 0.74 PDE4D (0.50) HTTALDH1A1GAAKDM4ENPC1
SCHEMBL32674134 0.74 MAPT (0.59) ADORA2AADORA1ALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187923-A 2 aryl 4 aroyl triazole compounds and application thereof 沈阳药科大学 2016-12-07 CN disclosed