SCHEMBL28091089

SCHEMBL28091089

C#Cc1cc(C)cc(C)c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 6/20 0.40
TSHR P16473 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
RAPGEF4 Q8WZA2 5/20 0.39
LMNA P02545 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HSD17B10 Q99714 1/20 0.35
POLB P06746 2/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
PTPN1 P18031 1/20 0.32
PTPN6 P29350 1/20 0.32
PTPN11 Q06124 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
NUDT1 P36639 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16727104 0.80 KDM4E (0.34) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL6152098 0.79 KDM4E (0.45) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL6589859 0.79 KDM4E (0.41) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL16128805 0.77 ALDH1A1 (0.37) ALDH1A1TSHRTDP1TP53CYP3A4
SCHEMBL139002 0.76 ALDH1A1 (0.65) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL3704142 0.74 ALDH1A1 (0.34) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL30578150 0.73 ALDH1A1 (0.61) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL28908462 0.73 ALDH1A1 (0.61) KDM4EALDH1A1TSHRTDP1TP53
Methane SCHEMBL2038793 0.73 ALDH1A1 (0.61) KDM4EALDH1A1TSHRTDP1TP53
SCHEMBL30578152 0.73 ALDH1A1 (0.61) KDM4EALDH1A1TSHRTDP1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105859725-B The synthetic method of 5,10 indoline simultaneously [3,2 b] indole derivatives 天津大学 2017-11-17 CN disclosed
CN-105859725-A 5,10-dihydroindolo[3,2-b]indole derivative synthesis method 天津大学 2016-08-17 CN disclosed