SCHEMBL28091184

SCHEMBL28091184

COOC(=O)c1ccc2scnc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
KDM4E B2RXH2 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
HKDC1 Q2TB90 1/20 0.46
NAMPT P43490 1/20 0.46
ESR1 P03372 2/20 0.45
CRBN Q96SW2 2/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HSD11B1 P28845 1/20 0.43
NTRK1 P04629 2/20 0.42
NTRK2 Q16620 2/20 0.42
CLK1 P49759 1/20 0.42
CLK2 P49760 1/20 0.42
CLK3 P49761 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19900857 0.88 NPC1 (0.62) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL29852002 0.88 NAMPT (0.51) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL1538274 0.88 NAMPT (0.51) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL260218 0.84 SMN1; SMN2 (0.51) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL31266420 0.84 SMN1; SMN2 (0.51) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL8861663 0.79 NPC1 (0.53) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL5279767 0.78 NAMPT (0.46) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL11507433 0.78 ESR1 (0.52) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL30917341 0.77 NPC1 (0.74) NPC1RAB9AKDM4EL3MBTL1TDP1
SCHEMBL261022 0.77 NPC1 (0.74) NPC1RAB9AKDM4EL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103524559-B Ester derivant of polysubstituted 4-methylamino benzenecarboximidamide and its production and use 西藏海思科药业集团股份有限公司 2016-09-28 CN disclosed