SCHEMBL28092572

SCHEMBL28092572

O=C(OCCC(F)(F)F)N1CCNc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 5/20 0.44
HSD11B1 P28845 2/20 0.40
MAPK1 P28482 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
GAA P10253 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
THRB P10828 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
GPBAR1 Q8TDU6 2/20 0.37
HSD17B3 P37058 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TACR1 P25103 1/20 0.34
AVPR2 P30518 1/20 0.33
IDH1 O75874 1/20 0.33
BCHE P06276 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
HTR1A P08908 1/20 0.33
CHRM5 P08912 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28092694 0.87 AVPR1A (0.45) AVPR1AHSD11B1MAPK1NPC1RAB9A
SCHEMBL3094477 0.81 AVPR1A (0.55) AVPR1AHSD11B1MAPK1NPC1RAB9A
SCHEMBL9226464 0.81 BCHE (0.49) AVPR1AHSD11B1MAPK1NPC1RAB9A
SCHEMBL30379140 0.81 BCHE (0.49) AVPR1AHSD11B1MAPK1NPC1RAB9A
SCHEMBL28092454 0.77 HSD11B1 (0.46) AVPR1AHSD11B1MAPK1NPC1RAB9A
SCHEMBL28092508 0.77 P2RX4 (0.49) AVPR1AHSD11B1MAPK1NPC1RAB9A
SCHEMBL19949852 0.76 AVPR1A (0.51) AVPR1AHSD11B1MAPK1THRBGPBAR1
SCHEMBL29505992 0.75 MAPK1 (0.60) AVPR1AHSD11B1MAPK1THRBGPBAR1
SCHEMBL975814 0.75 MAPK1 (0.60) AVPR1AHSD11B1MAPK1THRBGPBAR1
SCHEMBL28092562 0.73 AVPR1A (0.49) AVPR1AHSD11B1MAPK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029076-A Benzopiperazine compositions as BET bromodomain inhibitors 福马疗法公司 2016-10-12 CN claimed
CN-106029076-A Benzopiperazine compositions as BET bromodomain inhibitors 福马疗法公司 2016-10-12 CN disclosed