SCHEMBL28092562

SCHEMBL28092562

O=C(Oc1ccccc1)N1CCNc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 2/20 0.49
GAA P10253 2/20 0.46
HSD11B1 P28845 1/20 0.44
BCHE P06276 1/20 0.43
ALDH1A1 P00352 3/20 0.42
GPBAR1 Q8TDU6 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
CHRNA7 P36544 1/20 0.40
HTR3A P46098 1/20 0.40
HSD17B3 P37058 1/20 0.40
MGLL Q99685 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MAPK1 P28482 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
AVPR2 P30518 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28092466 0.89 BCHE (0.48) AVPR1AHSD11B1BCHEGPBAR1
SCHEMBL28833120 0.89 AVPR1A (0.51) AVPR1AHSD11B1BCHEALDH1A1GPBAR1
SCHEMBL28092460 0.89 AVPR1A (0.45) AVPR1AGAAHSD11B1ALDH1A1GPBAR1
SCHEMBL28833101 0.87 HSD11B1 (0.44) AVPR1AGAAHSD11B1ALDH1A1GPBAR1
SCHEMBL28092698 0.86 BCHE (0.51) AVPR1AHSD11B1BCHEALDH1A1GPBAR1
SCHEMBL28092473 0.86 BCHE (0.51) AVPR1AHSD11B1BCHEALDH1A1GPBAR1
SCHEMBL28092682 0.86 AVPR1A (0.43) AVPR1AGAAHSD11B1ALDH1A1GPBAR1
SCHEMBL28092729 0.85 MGLL (0.48) ALDH1A1SMN1; SMN2MGLL
SCHEMBL28092668 0.84 MGLL (0.51) AVPR1AALDH1A1MGLLCYP3A4TSHR
SCHEMBL28092670 0.83 TRPV1 (0.46) AVPR1AGAAALDH1A1GPBAR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029076-A Benzopiperazine compositions as BET bromodomain inhibitors 福马疗法公司 2016-10-12 CN disclosed