SCHEMBL28096085

SCHEMBL28096085

NC(=O)c1nc(Cl)c2ccccc2n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.52
GRM2 Q14416 8/20 0.46
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
METAP1 P53582 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
GBA1 P04062 1/20 0.41
LCK P06239 1/20 0.41
MAP2K3 P46734 1/20 0.41
MAP2K6 P52564 1/20 0.41
BTK Q06187 1/20 0.41
MAP3K19 Q56UN5 1/20 0.41
NEK10 Q6ZWH5 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
PRNP P04156 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22694433 0.85 MAOA (0.47) MAOAMAOBMETAP1NCOA1KMT2A
SCHEMBL27845960 0.85 MAOA (0.47) MAOAMAOBMETAP1TP53ATM
SCHEMBL20352582 0.84 MAOA (0.45) MAOAMAOBMETAP1KMT2AATM
Hydrochloric Acid SCHEMBL14842653 0.79 DCPS (0.53) SCN9AMAOALCKMAP2K3MAP2K6
SCHEMBL14358666 0.79 HSD17B10 (0.59) SCN9AGRM2GBA1TP53KMT2A
SCHEMBL31413901 0.79 SCN9A (0.52) SCN9AGRM2MAOANCOA1NCOA3
SCHEMBL526900 0.78 KDM4E (0.57) GBA1TP53KMT2AKDM4E
Hydrochloric Acid SCHEMBL14842831 0.77 HSD17B10 (0.58) SCN9AGRM2GBA1TP53KMT2A
SCHEMBL10986022 0.77 SCN9A (0.76) SCN9AKMT2A
Bicarbonate SCHEMBL11023181 0.76 MAOA (0.48) MAOAMAOBMETAP1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008373-B Disubstituted bicyclic derivative and its application as efflux pump inhibitor in antibacterial 山东大学 2019-02-22 CN disclosed
CN-106008373-A Disubstituted bicyclic derivative and application thereof as efflux pump inhibitor to anti-microbial 山东大学 2016-10-12 CN disclosed