SCHEMBL28097302

SCHEMBL28097302

O=C(O)c1cccc(CN2CN=Cc3ccccc32)c1F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.42
SIRT1 Q96EB6 2/20 0.40
TTR P02766 1/20 0.36
MRGPRX4 Q96LA9 6/20 0.36
FABP3 P05413 1/20 0.35
FABP4 P15090 1/20 0.35
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
TRPA1 O75762 1/20 0.34
CACNA1G O43497 1/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28097260 0.87 BRD4 (0.41) BRD4SIRT1ALDH1A1ALOX15TRPA1
SCHEMBL28097306 0.74 PTGER4 (0.39) TTRMRGPRX4ALDH1A1
SCHEMBL28097300 0.74 ALDH1A1 (0.39) BRD4SIRT1ALDH1A1SIRT2
SCHEMBL31227713 0.69 MRGPRX4 (0.42) MRGPRX4FABP3ALDH1A1
SCHEMBL1645358 0.69 ALDH1A1 (0.50) MRGPRX4FABP3FABP4ALDH1A1
SCHEMBL28234956 0.67 P2RX4 (0.34) ALDH1A1
SCHEMBL27762359 0.67 KDM4E (0.40) ALDH1A1ALOX15
SCHEMBL30701130 0.67 ALDH1A1 (0.48) MRGPRX4ALDH1A1ALOX15
SCHEMBL1401459 0.66 MRGPRX4 (0.49) MRGPRX4ALDH1A1ALOX15
SCHEMBL4238088 0.66 KAT6A (0.54) MRGPRX4ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104230827-B 1-(aryl methyl) quinazoline-2,4 (1H, 3H)-diketone is as PARP inhibitor and application thereof 南京英派药业有限公司 2016-10-26 CN disclosed