SCHEMBL28097306

SCHEMBL28097306

O=C(O)c1cc(F)cc(CN2CN=Cc3ccccc32)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 3/20 0.39
PTGER2 P43116 3/20 0.39
KMT2A Q03164 1/20 0.34
PTGER1 P34995 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HCAR1 Q9BXC0 1/20 0.33
P2RY14 Q15391 1/20 0.33
REN P00797 1/20 0.33
CTSD P07339 1/20 0.33
CTSE P14091 1/20 0.33
KCNH2 Q12809 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
TTR P02766 1/20 0.33
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22042030 0.77 EPHX2 (0.40) KMT2ACYP2D6CYP2C9ALDH1A1
SCHEMBL28097300 0.74 ALDH1A1 (0.39) KMT2AP2RY14KCNH2DRD2CYP2D6
SCHEMBL28097302 0.74 BRD4 (0.42) MRGPRX4TTRALDH1A1
SCHEMBL7603456 0.71 KMT2A (0.40) KMT2ACYP2D6CYP2C9KDM4EALDH1A1
SCHEMBL31752008 0.70 KMT2A (0.68) KMT2AHDAC1ALDH1A1
SCHEMBL28149958 0.69 TYMS (0.41) KMT2ACYP2D6CYP2C9KDM4E
SCHEMBL28321833 0.68 PARP1 (0.51)
SCHEMBL28097260 0.68 BRD4 (0.41) KMT2ACYP2D6ALDH1A1
SCHEMBL31038288 0.66 AKR1B1 (0.40) KMT2AHDAC1HDAC6KDM4EALDH1A1
SCHEMBL28234956 0.66 P2RX4 (0.34) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104230827-B 1-(aryl methyl) quinazoline-2,4 (1H, 3H)-diketone is as PARP inhibitor and application thereof 南京英派药业有限公司 2016-10-26 CN disclosed