SCHEMBL28097333

SCHEMBL28097333

COc1cc(C(=O)OC(C)=O)cc(Br)c1OC

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.64
APOBEC3A P31941 1/20 0.64
HTT P42858 1/20 0.64
APOBEC3G Q9HC16 1/20 0.64
PTPN1 P18031 2/20 0.50
TNFRSF1A P19438 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 2/20 0.49
HPGD P15428 1/20 0.49
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.45
TPMT P51580 1/20 0.45
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7123362 0.88 MEN1 (0.56) TSHRHTTSMN1; SMN2LMNAKMT2A
SCHEMBL31520156 0.85 TSHR (0.70) TSHRAPOBEC3AHTTAPOBEC3GPTPN1
SCHEMBL30740936 0.85 TSHR (0.70) TSHRAPOBEC3AHTTAPOBEC3GPTPN1
SCHEMBL1134614 0.83 TSHR (0.72) TSHRAPOBEC3AHTTAPOBEC3GPTPN1
SCHEMBL10672750 0.81 TPMT (0.55) TSHRAPOBEC3AHTTAPOBEC3GPTPN1
SCHEMBL1204414 0.80 HTT (0.72) TSHRAPOBEC3AHTTAPOBEC3GTNFRSF1A
SCHEMBL30740894 0.80 HTT (0.72) TSHRAPOBEC3AHTTAPOBEC3GTNFRSF1A
SCHEMBL8430188 0.79 TSHR (0.66) TSHRAPOBEC3AHTTAPOBEC3GPTPN1
SCHEMBL8148063 0.79 MEN1 (0.61) TSHRAPOBEC3AHTTAPOBEC3GSMN1; SMN2
SCHEMBL985701 0.78 TSHR (0.70) TSHRAPOBEC3AHTTAPOBEC3GPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106278941-A Nine kinds of PTP1B inhibitor and synthesis thereof and application 南通中国科学院海洋研究所海洋科学与技术研究发展中心 2017-01-04 CN claimed