SCHEMBL28097825

SCHEMBL28097825

O=C(O)CCc1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.57
ITGB1 P05556 12/20 0.56
ITGA4 P13612 11/20 0.56
ITGA2 P17301 1/20 0.56
ITGB7 P26010 1/20 0.56
JAK2 O60674 1/20 0.55
CYP3A4 P08684 1/20 0.55
JAK1 P23458 1/20 0.55
TYK2 P29597 1/20 0.55
TAS1R3 Q7RTX0 1/20 0.55
TAS1R1 Q7RTX1 1/20 0.55
TAS1R2 Q8TE23 1/20 0.55
KMT2A Q03164 1/20 0.54
NR1H4 Q96RI1 1/20 0.53
ITGB3 P05106 1/20 0.52
ITGAV P06756 1/20 0.52
ITGA2B P08514 1/20 0.52
ITGB5 P18084 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6514115 0.86 ITGB1 (0.65) FFAR1ITGB1ITGA4NR1H4
SCHEMBL28097862 0.85 JAK2 (0.51) ITGB1ITGA4ITGA2ITGB7JAK2
SCHEMBL6601710 0.81 TYK2 (0.61) ITGB1ITGA4ITGA2ITGB7JAK2
SCHEMBL6930314 0.81 TYK2 (0.54) FFAR1ITGB1ITGA4ITGA2ITGB7
SCHEMBL5660001 0.79 LMNA (0.63) FFAR1NR1H4
SCHEMBL27515653 0.79 ITGB1 (0.64) ITGB1ITGA4ITGA2ITGB7ITGB3
SCHEMBL5230799 0.79 ITGB1 (0.64) ITGB1ITGA4ITGA2ITGB7ITGB3
SCHEMBL4154853 0.79 TYK2 (0.71) JAK2CYP3A4JAK1TYK2TAS1R3
SCHEMBL27581014 0.79 FFAR1 (0.59) FFAR1NR1H4
SCHEMBL1232960 0.78 NR1H4 (0.71) FFAR1ITGB1KMT2ANR1H4ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104023751-B Targeted delivery extremely expresses the integrin antagonists conjugate of the cell of VLA-4 弗·哈夫曼-拉罗切有限公司 2016-11-09 CN disclosed