SCHEMBL28097863

SCHEMBL28097863

CC(C)C(=O)Oc1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 3/20 0.52
JAK2 O60674 1/20 0.52
CYP3A4 P08684 1/20 0.52
JAK1 P23458 1/20 0.52
TAS1R3 Q7RTX0 2/20 0.52
TAS1R1 Q7RTX1 2/20 0.52
TAS1R2 Q8TE23 1/20 0.52
KMT2A Q03164 2/20 0.51
GAA P10253 2/20 0.47
MAPT P10636 1/20 0.47
RAB9A P51151 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ITGB1 P05556 6/20 0.47
ITGA4 P13612 6/20 0.47
ELANE P08246 2/20 0.46
TLR8 Q9NR97 2/20 0.46
TLR7 Q9NYK1 2/20 0.46
ITGA2 P17301 1/20 0.46
ITGB7 P26010 1/20 0.46
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6509781 0.80 KLK7 (0.44) TYK2JAK2CYP3A4JAK1TAS1R3
SCHEMBL16677947 0.78 ELANE (0.57) TAS1R3TAS1R1TAS1R2KMT2AGAA
SCHEMBL6679298 0.78 KMT2A (0.49) CYP3A4KMT2AMAPTITGB1ITGA4
SCHEMBL6509892 0.78 CNR2 (0.46) KMT2AMAPTITGB1ITGA4ALDH1A1
Hydrochloric Acid SCHEMBL6514192 0.77 TYK2 (0.51) TYK2JAK2CYP3A4JAK1TAS1R3
SCHEMBL7384072 0.76 TYK2 (0.65) TYK2JAK2CYP3A4JAK1TAS1R3
SCHEMBL4154853 0.73 TYK2 (0.71) TYK2JAK2CYP3A4JAK1TAS1R3
SCHEMBL25219057 0.73 TYK2 (0.66) TYK2TAS1R3TAS1R1TAS1R2KMT2A
SCHEMBL16677858 0.73 LMNA (0.56) CYP3A4KMT2AGAAMAPTRAB9A
SCHEMBL16675163 0.73 LMNA (0.60) CYP3A4KMT2AGAAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104023751-B Targeted delivery extremely expresses the integrin antagonists conjugate of the cell of VLA-4 弗·哈夫曼-拉罗切有限公司 2016-11-09 CN disclosed