Dimethyl Maleate

Dimethyl Maleate

SCHEMBL28099231

C=CC(=O)OCCO.COC(=O)/C=C\C(=O)OC

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Dimethyl Maleate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.50
TSHR P16473 7/20 0.73
HCAR2 Q8TDS4 5/20 0.50
ALDH1A1 P00352 4/20 0.50
TP53 P04637 3/20 0.50
HIF1A Q16665 3/20 0.50
CYP3A4 P08684 2/20 0.50
NFE2L2 Q16236 1/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
THRB P10828 2/20 0.42
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ATM Q13315 1/20 0.39
ACHE P22303 1/20 0.34
MAPT P10636 2/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
GFPT1 Q06210 1/20 0.34
CACNA1B Q00975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Monomethyl Fumarate SCHEMBL28099233 0.93 TSHR (0.63) TSHRHCAR2ALDH1A1TP53HIF1A
Acrylic Acid Methyl Ester SCHEMBL6374663 0.92 TSHR (0.79) TSHRHCAR2ALDH1A1TP53HIF1A
SCHEMBL8894920 0.88 TSHR (0.59) TSHRHCAR2ALDH1A1TP53HIF1A
SCHEMBL12310431 0.88 TSHR (0.59) TSHRHCAR2ALDH1A1TP53HIF1A
SCHEMBL7262708 0.88 HCAR2 (0.59) TSHRHCAR2ALDH1A1KEAP1NFE2L2
SCHEMBL2980459 0.88 HCAR2 (0.59) TSHRHCAR2ALDH1A1KEAP1NFE2L2
SCHEMBL2980456 0.88 HCAR2 (0.59) TSHRHCAR2ALDH1A1KEAP1NFE2L2
Methoxymethane SCHEMBL863787 0.88 TSHR (0.86) TSHRHCAR2ALDH1A1TP53HIF1A
Acrylic Acid Methyl Ester SCHEMBL4866248 0.87 TSHR (0.70) TSHRHCAR2ALDH1A1TP53HIF1A
SCHEMBL4147710 0.86 TSHR (0.83) TSHRHCAR2ALDH1A1TP53HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102844401-B Expandable elastomeric material in the presence of water or oil 罗地亚管理公司 2016-08-31 CN claimed