Monomethyl Fumarate

Monomethyl Fumarate

SCHEMBL28099233

C=CC(=O)OCCO.COC(=O)/C=C\C(=O)O

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Monomethyl Fumarate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.43
TSHR P16473 6/20 0.63
HCAR2 Q8TDS4 9/20 0.57
HPGD P15428 1/20 0.44
ALDH1A1 P00352 6/20 0.44
TP53 P04637 3/20 0.44
HIF1A Q16665 3/20 0.44
HSD17B10 Q99714 2/20 0.44
CYP3A4 P08684 2/20 0.44
NFE2L2 Q16236 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALOX15 P16050 1/20 0.40
RECQL P46063 1/20 0.40
THRB P10828 2/20 0.38
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethyl Maleate SCHEMBL28099231 0.93 TSHR (0.73) TSHRHCAR2HPGDALDH1A1TP53
SCHEMBL29132468 0.90 TSHR (0.73) TSHRHCAR2HPGDALDH1A1TP53
Fumaric Acid SCHEMBL956152 0.89 TSHR (0.79) TSHRHCAR2HPGDALDH1A1TP53
Maleic Acid SCHEMBL956148 0.89 TSHR (0.79) TSHRHCAR2HPGDALDH1A1TP53
Fumaric Acid SCHEMBL30592706 0.89 TSHR (0.79) TSHRHCAR2HPGDALDH1A1TP53
Acrylic Acid Methyl Ester SCHEMBL4866248 0.88 TSHR (0.70) TSHRHCAR2HPGDALDH1A1TP53
Acrylic Acid Methyl Ester SCHEMBL6374663 0.86 TSHR (0.79) TSHRHCAR2HPGDALDH1A1TP53
SCHEMBL29185571 0.83 TSHR (0.63) TSHRHCAR2HPGDALDH1A1TP53
Crotonic Acid SCHEMBL9681122 0.83 TSHR (0.68) TSHRHCAR2HPGDALDH1A1TP53
Crotonic Acid SCHEMBL9681135 0.83 TSHR (0.68) TSHRHCAR2HPGDALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102844401-B Expandable elastomeric material in the presence of water or oil 罗地亚管理公司 2016-08-31 CN claimed