SCHEMBL28103418

SCHEMBL28103418

COc1ccc(Cc2c(C)nn(C)c2Nc2c(F)cccc2Br)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
P2RX7 Q99572 3/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
KMT2A Q03164 2/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CHRM4 P08173 1/20 0.32
TP53 P04637 1/20 0.32
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28103412 0.92 P2RX7 (0.38) PDE4APDE4BPDE4CPDE4DP2RX7
SCHEMBL28103211 0.91 PDE4A (0.33) PDE4APDE4BPDE4CPDE4DP2RX7
SCHEMBL28835079 0.88 P2RX7 (0.38) P2RX7KDM4EPOLBKMT2ASMN1; SMN2
SCHEMBL28103627 0.87 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DP2RX7
SCHEMBL28103422 0.81 RXFP1 (0.36) PDE4APDE4BPDE4CPDE4DP2RX7
SCHEMBL173457 0.81 POLB (0.39) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL28103433 0.79 RXFP1 (0.36) PDE4APDE4BPDE4CPDE4DP2RX7
SCHEMBL173247 0.77 CRHR1 (0.40) POLBKMT2AGAAMAPK1SMN1; SMN2
SCHEMBL170536 0.74 POLB (0.38) KDM4EPOLBGAAMAPK1TP53
SCHEMBL28835063 0.72 RXFP1 (0.39) PDE4APDE4BPDE4CPDE4DP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106417305-A Fungicidal pyrazoles and their mixtures 杜邦公司 2017-02-22 CN claimed
CN-106417305-A Fungicidal pyrazoles and their mixtures 杜邦公司 2017-02-22 CN disclosed
CN-106008299-A Intermediate for preparing fungicidal pyrazoles 杜邦公司 2016-10-12 CN disclosed