SCHEMBL28104875

SCHEMBL28104875

CN1CCC(n2cc(N)cn2)C1.Cc1cc(C(=O)O)cc(C(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 2/20 0.44
TPMT P51580 1/20 0.39
KDM2B Q8NHM5 2/20 0.38
NAMPT P43490 1/20 0.36
ALOX15 P16050 1/20 0.35
MELK Q14680 2/20 0.35
DYRK1A Q13627 6/20 0.34
GSK3B P49841 5/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34
MAPK7 Q13164 1/20 0.34
ALDH1A1 P00352 1/20 0.34
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
RORC P51449 1/20 0.33
MET P08581 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23685815 0.83 KDM5A (0.47) KDM5ANAMPTALOX15MELKFLT4
SCHEMBL9953033 0.83 KDM5A (0.47) KDM5ANAMPTALOX15MELKFLT4
SCHEMBL31361718 0.83 KDM5A (0.47) KDM5ANAMPTALOX15MELKFLT4
SCHEMBL27660981 0.77 KDM2B (0.40) TPMTKDM2BDYRK1AGSK3BCLK2
SCHEMBL17076683 0.75 KDM5A (0.43) KDM5AALOX15MELK
SCHEMBL531181 0.75 KDM5A (0.43) KDM5AALOX15MELK
SCHEMBL216558 0.74 ALOX15 (0.50) KDM5AALOX15DYRK1AGSK3BCLK2
SCHEMBL14706020 0.73 ACHE (0.48) MELKDYRK1AGSK3BCLK2CLK3
Hydrochloric Acid SCHEMBL15145595 0.73 ALOX15 (0.49) KDM5AALOX15DYRK1AGSK3BCLK2
SCHEMBL12093350 0.73 OGA (0.43) KDM5AALOX15MELKFLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105940004-A Compounds 葛兰素史密斯克莱知识产权发展有限公司 2016-09-14 CN disclosed