SCHEMBL28107101

SCHEMBL28107101

CS(=O)(=O)c1ccc(-c2ncccc2[N+](=O)[O-])cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.58
PTGS1 P23219 2/20 0.58
PAX8 Q06710 1/20 0.54
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
RAB9A P51151 1/20 0.52
TRPV1 Q8NER1 1/20 0.51
PDE10A Q9Y233 1/20 0.44
MAPT P10636 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ERN1 O75460 1/20 0.43
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
HSD11B1 P28845 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28106815 0.86 MEN1 (0.51) PTGS2PTGS1PAX8MEN1KMT2A
SCHEMBL1736457 0.83 PAX8 (0.57) PAX8MEN1KMT2ARAB9ATRPV1
SCHEMBL444703 0.80 ALDH1A1 (0.53) PTGS2PTGS1MEN1KMT2ARAB9A
SCHEMBL1736168 0.80 MEN1 (0.57) MEN1KMT2ARAB9ATRPV1PDE10A
SCHEMBL1738384 0.80 MAPT (0.52) MEN1KMT2ARAB9ATRPV1PDE10A
SCHEMBL27930436 0.80 TRPV1 (0.51) PAX8MEN1KMT2ARAB9ATRPV1
SCHEMBL28567279 0.79 PDE10A (0.50) PAX8MEN1KMT2ARAB9ATRPV1
SCHEMBL1738423 0.79 NPC1 (0.56) MEN1KMT2ARAB9ATRPV1PDE10A
SCHEMBL1735377 0.79 TRPV1 (0.51) PAX8MEN1KMT2ARAB9ATRPV1
SCHEMBL31451585 0.79 NPC1 (0.56) MEN1KMT2ARAB9ATRPV1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029663-A Tricyclic compounds as anticancer agents 百时美施贵宝公司 2016-10-12 CN disclosed