SCHEMBL2810876

SCHEMBL2810876

CCOC(=O)c1[nH]c2ccccc2c1-c1ccc(C(C)(C)C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
HPGD P15428 4/20 0.58
CYP1A2 P05177 1/20 0.58
XBP1 P17861 1/20 0.58
CYP2C19 P33261 1/20 0.58
KDM4E B2RXH2 9/20 0.56
TSHR P16473 1/20 0.54
HSD17B10 Q99714 1/20 0.54
HTR6 P50406 2/20 0.53
TUBB4A P04350 2/20 0.52
TUBB P07437 2/20 0.52
TUBA3C P0DPH7 2/20 0.52
TUBA1B P68363 2/20 0.52
TUBA4A P68366 2/20 0.52
TUBB4B P68371 2/20 0.52
TUBB3 Q13509 2/20 0.52
TUBB2A Q13885 2/20 0.52
TUBB8 Q3ZCM7 2/20 0.52
TUBA3E Q6PEY2 2/20 0.52
TUBA1A Q71U36 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13168431 0.89 ALDH1A1 (0.51) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL2956667 0.87 ALDH1A1 (0.73) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL2809161 0.87 ALDH1A1 (0.48) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL7679486 0.85 ALDH1A1 (0.60) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL7673201 0.85 ALDH1A1 (0.74) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL6857725 0.84 HPGD (0.62) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL7560870 0.83 HPGD (0.56) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL7676091 0.83 ALDH1A1 (0.58) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL7528226 0.82 ALDH1A1 (0.60) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL24074728 0.82 ALDH1A1 (0.57) ALDH1A1HPGDCYP1A2XBP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11077421-B2 Carbon sorbent for removal of metal catalysts from pharmaceuticals TDA RESEARCH, INC. (US) 2021-08-03 US disclosed
US-20190099737-A1 CARBON SORBENT FOR REMOVAL OF METAL CATALYSTS FROM PHARMACEUTICALS TDA RESEARCH, INC. 2019-04-04 US disclosed
WO-2017172512-A1 CARBON SORBENT FOR REMOVAL OF METAL CATALYSTS FROM PHARMACEUTICALS TDA RESEARCH, INC. (US) 2017-10-05 WO disclosed
US-20100240642-A1 1H-Indole-2-Carboxylic Acid Derivatives Useful As PPAR Modulators SMITHKLINE BEECHAM CORPORATION (US) 2010-09-23 US disclosed
EP-2081894-A1 1H-INDOLE-2-CARBOXYLIC ACID DERIVATIVES USEFUL AS PPAR MODULATORS SmithKline Beecham Corporation (US) 2009-07-29 EP disclosed
WO-2008028118-A1 1H-INDOLE-2-CARBOXYLIC ACID DERIVATIVES USEFUL AS PPAR MODULATORS SMITHKLINE BEECHAM CORPORAITON (US) 2008-03-06 WO disclosed
US-6787651-B2 2-CARBOXY-SUBSTITUTED; TREATING OSTEOPENIA, OSTEOPOROSIS, CANCER, DIABETES AND ATHEROSCLEROSIS. SMITHKLINE BEECHAM CORPORATION 2004-09-07 US disclosed
EP-1341761-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2003-09-10 EP disclosed
US-20030087902-A1 Substituted indoles, pharmaceutical compounds containing such indoles and their use as PPAR-gamma binding agents SMITHKLINE BEECHAM CORPORATION 2003-05-08 US disclosed
WO-2002030895-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-η BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11077421-B2 Carbon sorbent for removal of metal catalysts from pharmaceuticals RICTOR, SLC7A5, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 ALDH1A1 4287/4885HPGD 3105/4885CYP1A2 698/4885
US-20030087902-A1 Substituted indoles, pharmaceutical compounds containing such indoles and their use as PPAR-gamma binding agents PPARG, PPARA, PPARD ALDH1A1 2691/4885HPGD 442/4885CYP1A2 2218/4885
US-20100240642-A1 1H-Indole-2-Carboxylic Acid Derivatives Useful As PPAR Modulators PPARD, PPARA, PPARG ALDH1A1 402/4885HPGD 421/4885CYP1A2 216/4885
US-20190099737-A1 CARBON SORBENT FOR REMOVAL OF METAL CATALYSTS FROM PHARMACEUTICALS RICTOR, SLC7A5, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 ALDH1A1 4287/4885HPGD 3105/4885CYP1A2 698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.