SCHEMBL28110787

SCHEMBL28110787

Cc1ccc(Cl)c(C)c1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
HTT P42858 2/20 0.39
PTGS1 P23219 2/20 0.39
PTGS2 P35354 2/20 0.39
ADRA2A P08913 1/20 0.39
ADORA2A P29274 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP2A6 P11509 1/20 0.38
FABP3 P05413 1/20 0.37
FABP4 P15090 1/20 0.37
BRD4 O60885 2/20 0.37
AKT2 P31751 2/20 0.37
TDO2 P48775 1/20 0.37
KMT2A Q03164 1/20 0.37
PPARA Q07869 1/20 0.36
MAPT P10636 2/20 0.36
PLA2G7 Q13093 1/20 0.36
CYP1A2 P05177 1/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640023 1.00 ALDH1A1 (0.40) ALDH1A1HTTPTGS1PTGS2ADRA2A
SCHEMBL12925884 0.86 CYP2A6 (0.41) ALDH1A1HTTPTGS1PTGS2ADRA2A
SCHEMBL27930519 0.84 FABP3 (0.41) HTTPTGS1PTGS2ADRA2AADORA2A
SCHEMBL30159162 0.83 FABP3 (0.41) ALDH1A1HTTPTGS1PTGS2ADRA2A
SCHEMBL28999631 0.81 ESR2 (0.48) ALDH1A1HTTPTGS1PTGS2PPARA
SCHEMBL7649808 0.79 CYP1A2 (0.43) ALDH1A1PTGS1PTGS2HSD17B10CYP2A6
SCHEMBL27397239 0.79 SMN1; SMN2 (0.44) ALDH1A1HTTPTGS1PTGS2ADRA2A
SCHEMBL22391489 0.78 MAPT (0.48) ALDH1A1HTTPTGS1PTGS2HSD17B10
SCHEMBL28650275 0.77 IKBKB (0.46) ALDH1A1HSD17B10KMT2AMAPTCYP1A2
SCHEMBL23003867 0.77 POLB (0.46) ALDH1A1HTTPTGS1PTGS2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106132414-A Aryl lactams inhibitors of kinases 百时美施贵宝公司 2016-11-16 CN disclosed